Yohimbin hydrochloride 5mg #50

Yohimbin hydrochloride instruction

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Composition

One tablet of Yohimbin hydrochloride contains 5 mg of the same substance.
Excipients: lactose monohydrate, starch, hypromellose, calcium stearate, celactose.

Form of issue

Yohimbin hydrochloride hydrochloride is a tablet of white or pale yellow color. The drug is produced by 50 tablets in a plastic jar or polymer container; one such bank or container in a pack of paper.

pharmachologic effect

Stimulates potency.

Pharmacodynamics

Yohimbin hydrochloride enhances potency (aphrodisiac) and is an alkaloid derived from the bark of the Corynanthe tree.
The effect is due to selective inhibition of α2-adrenergic receptors. Activates adrenergic neurons in the brain, has a psychostimulating effect. It is likely that it also affects dopaminergic, serotonergic and cholinergic systems.
Yohimbin hydrochloride stimulates sexual behavior and restores reduced sexual activity and impaired erection due to stress.
The therapeutic effect is explained by the effects of Yohimbin hydrochloride hydrochloride, affecting the nervous system. Probably enhances the circulation of the penis and has a direct effect on the tissues involved in erection.

Pharmacokinetics

Completely absorbed in the intestine within an hour. The greatest concentration in the blood occurs in 40-70 minutes. When oral intake in the recommended doses of accumulation of the drug in the body does not occur. The half-life period depends on the dose taken.
82% Yohimbin hydrochloride binds to plasma proteins. Metabolised in the liver. Two main metabolites are known: active 11-hydroxyiodibimine and weakly active 10-hydroxy Yohimbin hydrochloride.

Indications for use

Therapy of functional and psychogenic impotence, male menopause, atony of the bladder.

Contraindications

    Hypersensitivity to Yohimbin or other components of the drug.
    Pronounced arterial hypotension.
    Severe liver and kidney damage.
    Therapy with adrenomimetics.
    This medication is not intended for use by women and children.

Side effects

    Cardiovascular disorders: tachycardia, increased pressure.
    Neurological disorders: tremor, dizziness, headache, sleep disturbance, excitability, sweating.
    Digestive system disorders: loss of appetite, nausea and vomiting, diarrhea.
    Reactions from the skin: hyperemia.
    Others: decreased diuresis, priapism, allergic reactions.

Instructions for use (Method and dosage)

Instruction prescribes to take the drug orally during meals, squeezed with water and not chewing. 1-2 tablets from one to three times a day.
The dose is recommended to be selected individually. The initial dose is 2.5 mg 3 times a day, the maximum dose is 1-2 tablets three times a day.
The effect in a number of cases occurs in a few weeks. The duration of therapy depends on the disease clinic and can be 4 weeks.

Overdose

Symptoms of peridosis. After 30-45 minutes after taking an excessive dose, generalized paresthesias develop, weakness, memory impairment, dizziness, headache, tremor, increased pressure, tachycardia, a sense of fear, increased norepinephrine in the blood, nausea, mydriasis, vomiting, sweating. These symptoms can persist for 2-3 hours.
Treatment: stop taking the drug, rinse the stomach, then take activated charcoal. As an antidote, Clonidine can be used that neutralizes mental effects and disorders of the sympathetic nervous system.
For the treatment of hypertensive crisis, β-adrenoblockers in combination with α-adrenoblockers or peripheral vasodilators are recommended. In case of an overdose it is forbidden to use neuroleptics with phenothiazine series.

Interaction

When combined with clonidine, the effects of drugs are mutually neutralized.
Clopyramine increases the concentration of Yohimbin hydrochloride hydrochloride in blood plasma.
Yohimbin hydrochloride enhances the action of antidepressants and increases the risk of developing side effects caused by them.
Joint reception with tranquilizers weakens the activity of the latter.

Storage conditions

    Store at a temperature of no higher than 25 degrees.
    Keep away from children.
Shelf life Three years.

special instructions

The formulation includes lactose and patients with galactose intolerance, glucose-galactose malabsorption syndrome, or lactase deficiency are prohibited from using this drug.

Yohimbin hydrochloride for weight loss

Sometimes the drug is used in sports nutrition, as a stimulator of the fat burning process (including in bodybuilding).

Therefore, there is often a question "how to take Yohimbin for weight loss?" It is believed that a safe dose is 10-20 mg, used separately with food in several receptions. However, doctors do not recommend taking this drug for other purposes because of possible side effects.

Reviews of Yohimbin hydrochloride

There are numerous positive reviews about Yohimbin hydrochloride, including when used for weight loss in bodybuilding and during sports. It should be remembered that before taking the drug should always consult with your doctor.