Clenbuterol Sopharma tabs 0.2mg #50

Clenbuterol Sopharma instruction for use

You can buy Clenbuterol on this page

Composition

1 tablet of pharmaceutical preparation Clenbuterol Sopharma contains such components as:
    Clenbuterol hydrochloride (basic biologically active substance) 0.2 mg;
    lactose monohydrate - 70 mg;
    microcrystalline cellulose (MCC) - 48.5 mg;
    wheat starch - 31.48 mg;
    Povidone To 25 - 6 mg;
    colloidal silicon dioxide - 2 mg;
    magnesium stearate - 2 mg.

Form of issue

In pharmacies, the drug can be found in the form:
    Tablets Clenbutrol 0.2 mg each. Filled in blisters (contour mesh packaging from aluminum foil or PVC) for 10 pieces. Cardboard packs, as a rule, contain 5 plates.

pharmachologic effect

The main component of the drug Klenbuterol Sopharma is selective beta2-adrenomimetic, that is, the mechanism of action of the biologically active component includes a stimulating effect on this type of receptors, which are mainly located in the bronchial tree. In response, the following cycle of secondary messengers is activated in the following sequence: Adenylate cyclase-cAMP-Protoninase A. Further, the effects of Clenbuterol extend to myosin, a component of smooth muscle fibers, which interacts with actin, and relaxes the bronchi. Thus, the problem of narrowing the lumen of the respiratory tract during the attacks of bronchial asthma is eliminated and respiratory processes are significantly facilitated.
Clenbuterol also has a secretolytic effect. In particular, the main component of the pharmaceutical preparation slows the release of inflammatory mediators and other active biological substances from mast cells, which increase bronchoconstriction. Due to these therapeutic properties, edema decreases, stagnant phenomena are eliminated in the lumen of the bronchial tree, mucociliary clearance is improved.
Separately, it should be noted the properties of Clenbuterol, which are used in sports pharmacology. The active component of the drug has anabolic properties like steroids, but it shows its effects with less force. The pharmaceutical is an active fat burner. The mechanism of this action is a slight increase in the internal temperature of the body, thereby increasing the consumption of calories. Among athletes and bodybuilders there is an opinion that an increase in temperature by 1 degree Celsius accelerates the metabolism of fats by 5 percent.
Thanks to such therapeutic effects, the stiffness of the muscular framework and the strength significantly exceed the initial readings before passing the conservative course. The body is given relief, venous and the desired appearance. Outwardly, such effects are comparable to a long-term low-calorie diet.

Pharmacodynamics and pharmacokinetics

The drug is used orally, after which it is sufficiently full and well absorbed from the gastrointestinal tract. Act Clenbuterol begins already after 10-15 minutes after ingestion, and the maximum therapeutic properties appear after 2-3 hours. Metabolized active components of the pharmaceutical drug in the liver, after which 78 percent of the metabolic products are excreted in the urine. An insignificant amount of metabolites is eliminated with bile in the lumen of the digestive tube.

Indications for use

    Bronchial asthma;
    Chronic obstructive pulmonary disease.

Contraindications

increased individual sensitivity to the components of the drug;
    acquired or hereditary intolerance of biologically active substances Clenbuterol Sopharma;
    tachycardia and tachyarrhythmia;
    thyrotoxicosis;
    idiopathic hypertrophic subaortic stenosis of the aorta;
    severe forms of coronary heart disease;
    acute period of myocardial infarction.
Conservative treatment of Clenbutrol against the background of the following pathologies should be conducted with caution, which implies therapy in special hospitals under the constant supervision of qualified medical personnel and conducting regular diagnostic tests:
    hyperthyroidism;
    diabetes;
    diseases of the cardiovascular system (in particular, severe arterial hypertension, cardiomyopathy, heart defects, ischemic disease or propensity to arrhythmias).

Side effects

    From the nervous system - headache and dizziness, anxiety, disturbance of sleep and wakefulness in the form of insomnia, intentional tremor of fingers.
    From the cardiovascular system - tachycardia, increased blood pressure, extrasystole, cardialgia.
    Gastrointestinal tract - dryness in the oral cavity, gastralgia, nausea, leading to vomiting.
    Local and generalized allergic reactions - urticaria, skin rash, bronchospasm, angioedema.
    From other systems of organs and tissues - muscle cramps, intense face hyperemia, increased sweating, hypokalemia and, as a result, muscle pain.
    There is the possibility of developing the "rebound" syndrome and resistance when the pharmaceutical product is canceled.
Separately, it should be noted the development of muscle cramps, when Clenbutrol in tablets is used by athletes and bodybuilders. This side effect is due to depletion of endogenous taurine reserves, deficiency of sodium and potassium electrolytes, and a general lack of water-salt metabolism. To facilitate muscle spasms, the following dietary changes are recommended:
    the use of an abundant amount of fruits (especially bananas, since they contain a lot of potassium);
    abundant drinking;
    additional inclusion of taurine in an amount of 3-5 grams per day;
    tableted potassium supplements daily before bedtime on an empty stomach (not less than 200-400 mg).

Tablets Clenbuterol, instructions for use (Method and dosage)

A syrup is given for oral administration. For adults, the optimal dosage is 15 ml 2-3 times a day at the beginning of a course of conservative treatment. After relieving the severe condition, the amount of prescribed medication should be reduced to a maintenance dose of 10 ml 2 times a day.
The instruction on the use of the pharmaceutical drug allows it to be used in pediatric practice, however, with strict adherence to the following dosages:
    children up to 8 months with a mass of 4-8 kg - 2.5 ml 2 times a day;
    from 8 months to 2 years (weighing about 8-12 kg) - 5 ml 2 times a day;
    age category from 2 to 4 years (12-16 kg) - 7.5 ml 2 times a day;
    children from 4 to 6 years and weight in the range of 16-22 kg - 10 ml 2 times a day;
    from 6 to 12 years (22-35 kg) - 15 ml 2 times a day;
    children over 12 years and weighing more than 35 kg - 15 ml 2-3 times a day.
Tablets, like syrup, are applied orally. The dosage of the pharmaceutical preparation depends on the body weight and the body's reaction in the form of side effects or adverse effects of the drug. The average amount of the drug used for men is about 100-140 μg, and for women 80-100 μg per day. Admission should not begin with the optimal dosage, but accumulate it gradually to provide the maximum therapeutic effect. That is, the conservative course starts with 1 tablet a day, and then increases by 1 tablet every day.
The duration of such therapy is about 8-10 weeks on average. However, a special drug regimen is used, since Clenbuterol does not have its anabolic effects after 18 days of continuous use. Therefore, the course consists of 2 weeks of continuous admission and 2 weeks of rest in turn, until the pharmaceutical product is over or the attending physician stops discontinuing its further use.

Overdose

The use of dosages that exceed the prescribed dosages is accompanied by:
    arrhythmia;
    tachycardia;
    gipolkalemia;
    arterial hypertension;
    tremor of extremities;
    pain in the heart.
There is no specific antidote for Clenbuterol, therefore detoxification and symptomatic therapy is used as treatment, that is, gastric lavage, the administration of oral sorbents (for example, activated carbon), the use of water-salt solutions for restoring the corresponding metabolic disorders, monitoring serum potassium levels and correction its proper way.

Interaction

When prescribing Clenbuterol Sopharm, the following clinical interactions of the pharmaceutical preparation should be considered:
    antagonism with the beta-blockers opposite in action;
    violation of intracardiac conductivity when combined with MAO inhibitors (monoamine oxidase) and Teofillin;
    a decrease in the effectiveness of the use of hypoglycemic agents (requires the recalculation of dosages for diabetes mellitus);
    an increase in the toxicity of cardiac glycosides (significantly increases the risk of developing a pathological condition, such as arrhythmia);
    Increase of own toxicity in combination with mimetics of sympathetic nature.

Storage conditions

Store the pharmaceutical product in a dark place, with a moderate humidity and at a temperature of no higher than 25 degrees Celsius. Also, medicinal tablets should be out of the reach of young children.
Shelf life - 3 years

special instructions

The adverse effects of conservative treatment with a pharmaceutical drug include intentional tremor, dizziness, weakness, therefore, during the course of the therapeutic course, one should refrain from performing potentially dangerous activities requiring maximum attention concentration and reaction speed. So, for example, you should not drive a car or other means of transportation yourself.

Children

The drug can be used in pediatric practice only in view of the above dosages, calculated for certain age categories and body weight of the child.

For losing weight

The drug can be used as a fat burner in sports pharmacology, since the active ingredients increase the body's internal temperature (see the explanation of the mechanism of action above).

During pregnancy (and lactation)

Clenbuterol in tablets has a tocolytic property to a certain extent, therefore, it is not necessary to prescribe a pharmaceutical product during the bearing of the child, during the prenatal and patrimonial periods. Absolutely contraindicated drug in the first trimester of pregnancy.
Clinical studies have not reliably confirmed or denied the fact that the active ingredient is able to enter breast milk. In the absence of relevant data, the administration of a pharmaceutical preparation is possible only if the expected beneficial therapeutic effect of the tablets is significantly greater than the potential risk to the child.

Reviews of Clenbuterol Sopharma

First of all, it should be noted that much more reviews about the pharmaceutical preparation, as a means to effectively kill spasm of the bronchial tree during attacks of bronchial asthma. This therapeutic effect is abundantly used in medicine and is confirmed by clinical studies of qualified specialists. Of course, the drug has certain side effects, but its effect develops within 10-15 minutes after ingestion, which makes it possible to eliminate the pathological condition that threatens life in the shortest possible time.
However, on thematic forums and Internet resources, there are also reviews about another field of application of Clenbuterol. Athletes and bodybuilders prefer to use this pharmaceutical drug, like diet pills or so-called "drying". With this task, as with the elimination of bronchospasm, the drug copes with a hurray, since at the base of this action lie quite justified mechanisms. However, the course is accompanied by severe side effects in the form of muscle cramps, because, as a rule, such patients tend to lose excess weight as quickly as possible.
Unequivocally, we can say that during the conservative course of taking the drug Clenbuterol Sopharma should clearly follow the instructions in the dosage. Thanks to such simple actions, you can save yourself from unnecessary suffering, going to the doctors and other adverse consequences.